Therapeutic Targets Database
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TTD Drug ID: DAP000065

Drug Information
NameCarteolol
SynonymsC06874; D07624; Prestwick0_000446; BSPBio_000492; CID2583; Prestwick3_000446; 5-[3-(tert-butylamino)-2-hydroxypropoxy]-3,4-dihydro-1H-quinolin-2-one; Carteolol Monohydrochloride; Carteololum [INN-Latin]; LS-142779; L000777; I14-8021; C16H24N2O3; Prestwick1_000446; 5-({3-[(1,1-dimethylethyl)amino]-2-hydroxypropyl}oxy)-3,4-dihydroquinolin-2(1H)-one; Carteolol (INN); 51781-21-6 (mono hydrochloride); DB00521; Carteolol [INN:BAN]; Carteolol HCl; AB00514682; AC1L1E05; 51781-06-7; Prestwick2_000446; CHEBI:3437; 2(1H)-Quinolinone, 5-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)-3,4-dihydro-; BPBio1_000542; NCGC00179541-01; CHEMBL839; CARTEOLOL; 5-[3-(tert-butylamino)-2-hydroxypropoxy]-3,4-dihydroquinolin-2(1H)-one; SPBio_002431; Carteololum; Oprea1_672850; BRD-A42167015-003-03-7; UNII-8NF31401XG
Trade NameCartrol; Ocupress; Teoptic; Arteolol; Arteoptic; Calte; Cartíž|abak; Carteol; Cartíž|ol; Cartrol; Elebloc; Endak; Glauteolol; Mikelan; Poenglaucol; Singlauc
CompanyCIBA Vision Sterile Mfg
IndicationHypertension
[ICD9: 401   ICD10: I10, I11, I12, I13, I15]
Approved    [1]
Structure

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InChI1S/C16H24N2O3/c1-16(2,3)17-9-11(19)10-21-14-6-4-5-13-12(14)7-8-15
(20)18-13/h4-6,11,17,19H,7-10H2,1-3H3,(H,18,20)
InChIKeyLWAFSWPYPHEXKX-UHFFFAOYSA-N
Canonical SMILESCC(C)(C)NCC(COC1=CC=CC2=C1CCC(=O)N2)O    
Therapeutic ClassAntihypertensive Agents
CAS NumberCAS 51781-06-7
FormulaC16H24N2O3
PubChem Compound IDCID 2583.
PubChem Substance IDSID 9091.
ChEBI3437;
SuperDrug ATC IDC07AA15; S01ED05
SuperDrug CAS ID051781067;
TargetBeta adrenergic receptorAgonist[2][3]
Ref 1Penbutolol and carteolol: two new beta-adrenergic blockers with partial agonism. J Clin Pharmacol. 1990 May;30(5):412-21. To Reference
Ref 2Partial agonistic effects of carteolol on atypical beta-adrenoceptors in the guinea pig gastric fundus. Jpn J Pharmacol. 2000 Nov;84(3):287-92. To Reference
Ref 3Effects of prolonged treatment with beta-adrenoceptor antagonist, carteolol on systemic and regional hemodynamics in stroke-prone spontaneously hypertensive rats. J Pharmacobiodyn. 1991 Feb;14(2):94-100. To Reference



 

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